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ACVR1

ACVR1,全稱為激活素A受體I型(Activin A receptor type I),也被稱為ALK-2。該蛋白主要參與骨骼、心臟、軟骨、神經(jīng)和生殖系統(tǒng)的發(fā)育和調(diào)節(jié)。ACVR1蛋白與骨形態(tài)發(fā)生蛋白(BMP)信號通路密切相關(guān),在疾病與健康中發(fā)揮著重要作用。例如,ACVR1基因突變會導(dǎo)致進(jìn)行性骨化性纖維發(fā)育不良(FOP),這是一種罕見的常染色體顯性遺傳病,主要特征為先天性雙側(cè)拇指畸形和全身軟組織的進(jìn)行性異位骨化。此外,ACVR1蛋白還在淋巴瘤的發(fā)生發(fā)展中發(fā)揮作用,研究表明PRC2抑制劑通過激活BMP-ACVR1信號通路抑制B細(xì)胞淋巴瘤生長。目前,針對ACVR1蛋白的藥物研發(fā)主要集中在FOP和淋巴瘤的治療上,例如ACVR1/ALK2和JAK1/2抑制劑莫洛替尼為原發(fā)性骨髓纖維化癥(PMF)帶來了顯著療效突破,而PRC2抑制劑則有望成為治療B細(xì)胞淋巴瘤的新選擇。

熱銷產(chǎn)品

ACVR1 Antibody (CSB-PA001257ESR2HU)

驗證數(shù)據(jù)

CSB-PA001257ESR2HU

Western blot
All lanes: ACVR1 antibody at 6μg/ml
Lane 1: A549 whole cell lysate
Lane 2: HepG2 whole cell lysate
Lane 3: Mouse gonad tissue
Secondary
Goat polyclonal to rabbit IgG at 1/10000 dilution
Predicted band size: 39 kDa
Observed band size: 39 kDa

CSB-PA001257ESR2HU

Immunohistochemistry of paraffin-embedded human kidney tissue using CSB-PA001257ESR2HU at dilution of 1:100

CSB-PA001257ESR2HU

Immunofluorescent analysis of PC-3 cells using CSB-PA001257ESR2HU at dilution of 1:100 and Alexa Fluor 488-congugated AffiniPure Goat Anti-Rabbit IgG(H+L)

ACVR1 Antibodies

ACVR1 for Homo sapiens (Human)

ACVR1 Proteins

ACVR1 Proteins for Rattus norvegicus (Rat)

ACVR1 Proteins for Mus musculus (Mouse)

ACVR1 Proteins for Bos taurus (Bovine)

ACVR1 Proteins for Gallus gallus (Chicken)